FundedIQ
Biotechnology

Septerna: Funding, Investors & Team (Oct 2026)

Septerna is a biotech firm focused on finding and developing groundbreaking small-molecule drugs that specifically target G protein-coupled receptors. By integrating cutting-edge small molecule drug discovery techniques with GPCR drug targets, Septerna aims to enhance patient well-being. Their Native Complex platform serves as the driving force behind these endeavors.

septerna.com LinkedIn San Francisco, United States 51-100 employees
Total raised
$150M
Rounds
1
Latest
Series B
Jul 2023

Septerna has raised $150M across 1 funding round on record, the most recent a Series B of $150M announced in Jul 2023.

That round is above the $8.4M median round size for Biotechnology companies tracked on FundedIQ over the last two years.

Septerna Company Profile and Key Stats

Total funding raised
$150M
across 1 round on record
Funding rounds on record
1
Latest funding round
Series B
$150M in Jul 2023
Employees
51-100
reported band
Headquarters
San Francisco, United States

Latest funding round on record: Jul 2023.

Septerna Funding Rounds

Date
Round
Amount
Series B
$150M

Septerna Founders and Leadership Team

Name
Role
Contact
Arthur Christopoulos
Founder
—

No contact details are on record for this team yet.

Septerna Funding Compared to Other Biotechnology Startups

Segment
Companies
Median round
4,185
$8.4M
30,319
$7.7M
4,422
$32M

Septerna's latest round of $150M is above the median round in Biotechnology. Medians cover the last 24 months of disclosed rounds.

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Septerna Funding FAQs

What does Septerna do?

Septerna is a biotech firm focused on finding and developing groundbreaking small-molecule drugs that specifically target G protein-coupled receptors. By integrating cutting-edge small molecule drug discovery techniques with GPCR drug targets, Septerna aims to enhance patient well-being. Their Native Complex platform serves as the driving force behind these endeavors.

How much funding has Septerna raised?

Septerna has raised $150M across 1 round on record. The most recent is a Series B of $150M announced in Jul 2023.

When did Septerna last raise funding?

Septerna's most recent funding round on record is a Series B of $150M, announced in Jul 2023.

Who founded Septerna?

FundedIQ lists Arthur Christopoulos (Founder) at Septerna.

Where is Septerna headquartered?

Septerna is based in San Francisco, California, United States.

How many employees does Septerna have?

Septerna is in the 51-100 employee band.

How does Septerna's funding compare to other Biotechnology startups?

Septerna's latest round of $150M is above the $8.4M median round size for Biotechnology companies on FundedIQ across 4,185 tracked companies over the last two years.

About FundedIQ's Septerna Funding Data

FundedIQ tracks announced funding rounds and refreshes this profile every week. Round dates, stages and amounts are normalised to a single format, converted to US dollars, and de-duplicated: two records of the same round announced days apart are merged, and two genuinely different rounds are kept apart on the amounts they disclose. Amounts shown are the disclosed figures only — a round announced without a number is listed and excluded from the total rather than estimated.

Employee counts are reported bands, not exact headcounts. Founder and executive names carry the job title on record. Anything we do not hold for Septerna is left off this page rather than filled in.

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